PDGs

 

The “druggable genome”, a term coined by Hopkins and Groom in 2002(3), defines a subset of genes in the human genome encoding proteins that may be amenable to modulation by drug-like molecules. To define potentially druggable genes (PDGs) in the human genome, we integrated the PDG candidates generated by six independent studies in which the druggable genes were systematically annotated by different strategies at a whole genome level. .

List of the PDGs in the human genome


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HGNC NameEnsembl Gene IDHGNC SymbolGenomic LocationTDLPubTator Score
relaxin 3ENSG00000171136RLN3chr19:14028148-14031042:+Tbio48.9376
interleukin 26ENSG00000111536IL26chr12:68201351-68225821:-Tbio33.8332
BCL2L2-PABPN1 readthroughENSG00000258643BCL2L2-PABPN1chr14:23306835-23325369:+0
solute carrier family 13 member 4ENSG00000164707SLC13A4chr7:135681237-135729258:-Tbio19.7576
phospholipase A2 group IVBENSG00000243708PLA2G4Bchr15:41837775-41848147:+Tchem0.883333
galanin receptor 3ENSG00000128310GALR3chr22:37823382-37825495:+Tchem17.3179
gamma-glutamyltransferase 2ENSG00000133475GGT2chr22:21207973-21227637:-Tbio0.833333
olfactory receptor family 2 subfamily T member 5ENSG00000203661OR2T5chr1:248488589-248489536:+Tdark12.875
urotensin 2 receptorENSG00000181408UTS2Rchr17:82374230-82375586:+Tchem85.7266
pregnancy specific beta-1-glycoprotein 1ENSG00000231924PSG1chr19:42866464-42879822:-Tbio3.58333
transmembrane phosphoinositide 3-phosphatase and tensin homolog 2ENSG00000132958TPTE2chr13:19422877-19536762:-Tbio11.3667
cyclin dependent kinase like 3ENSG00000006837CDKL3chr5:134286350-134371047:-Tchem6.18569
G protein-coupled receptor kinase 1ENSG00000185974GRK1chr13:113667155-113737735:+Tchem58.3694
solute carrier family 34 member 1ENSG00000131183SLC34A1chr5:177379235-177398848:+Tbio64.098
olfactory receptor family 7 subfamily A member 10ENSG00000127515OR7A10chr19:14840948-14841877:-Tdark0
chorionic somatomammotropin hormone 1ENSG00000136488CSH1chr17:63894909-63896661:-Tbio318.094
olfactory receptor family 2 subfamily L member 5ENSG00000197454OR2L5chr1:248021948-248022886:+Tdark0
olfactory receptor family 1 subfamily E member 2ENSG00000127780OR1E2chr17:3432870-3433841:-Tdark1
solute carrier family 41 member 3ENSG00000114544SLC41A3chr3:126006355-126101561:-Tdark1.58333
olfactory receptor family 1 subfamily D member 2ENSG00000184166OR1D2chr17:3092058-3092996:-Tbio36.6944

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