PDGs
The “druggable genome”, a term coined by Hopkins and Groom in 2002(3), defines a subset of genes in the human genome encoding proteins that may be amenable to modulation by drug-like molecules. To define potentially druggable genes (PDGs) in the human genome, we integrated the PDG candidates generated by six independent studies in which the druggable genes were systematically annotated by different strategies at a whole genome level. .
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HGNC Name | Ensembl Gene ID | HGNC Symbol | Genomic Location | TDL | PubTator Score |
chymotrypsinogen B2 | ENSG00000168928 | CTRB2 | chr16:75204096-75207185:- | Tchem | 8.03218 |
ribonuclease A family member 10 (inactive) | ENSG00000182545 | RNASE10 | chr14:20505537-20511169:+ | Tdark | 0.25 |
transglutaminase 6 | ENSG00000166948 | TGM6 | chr20:2380908-2432753:+ | Tchem | 31.1619 |
interferon alpha 21 | ENSG00000137080 | IFNA21 | chr9:21165637-21166660:- | Tbio | 10.9635 |
gamma-aminobutyric acid type A receptor subunit rho1 | ENSG00000146276 | GABRR1 | chr6:89177501-89231278:- | Tchem | 30.265 |
myosin light chain kinase 3 | ENSG00000140795 | MYLK3 | chr16:46703369-46790407:- | Tchem | 84.0718 |
G protein-coupled receptor 32 | ENSG00000142511 | GPR32 | chr19:50770464-50771732:+ | Tbio | 7.11905 |
potassium two pore domain channel subfamily K member 16 | ENSG00000095981 | KCNK16 | chr6:39314698-39322968:- | Tdark | 5.01069 |
hypocretin receptor 2 | ENSG00000137252 | HCRTR2 | chr6:55106460-55282620:+ | Tclin | 71.1857 |
olfactory receptor family 8 subfamily D member 4 | ENSG00000181518 | OR8D4 | chr11:123906146-123907476:+ | Tdark | 0 |
laeverin | ENSG00000172901 | LVRN | chr5:115962454-116027619:+ | Tbio | 15.3646 |
solute carrier family 4 member 9 | ENSG00000113073 | SLC4A9 | chr5:140360202-140375143:+ | Tbio | 10.8357 |
G protein-coupled receptor 12 | ENSG00000132975 | GPR12 | chr13:26755200-26760785:- | Tbio | 8.2381 |
olfactory receptor family 2 subfamily L member 3 | ENSG00000198128 | OR2L3 | chr1:248060682-248061620:+ | Tdark | 0 |
histatin 1 | ENSG00000126550 | HTN1 | chr4:70050402-70058845:+ | Tbio | 92.6583 |
UDP glucuronosyltransferase family 1 member A8 | ENSG00000242366 | UGT1A8 | chr2:233617645-233773310:+ | Tbio | 62.9186 |
parathyroid hormone 2 | ENSG00000142538 | PTH2 | chr19:49422414-49423441:- | Tdark | 34.4576 |
kelch like family member 10 | ENSG00000161594 | KLHL10 | chr17:41835685-41848384:+ | Tdark | 5.86667 |
integrin subunit alpha D | ENSG00000156886 | ITGAD | chr16:31393312-31426505:+ | Tbio | 17.4991 |
trace amine associated receptor 2 | ENSG00000146378 | TAAR2 | chr6:132617022-132624275:- | Tbio | 12.2917 |
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